Issue 56, 2015
From the journal:

Chemical Communications

Rh(iii)-catalyzed 7-azaindole synthesis via C–H activation/annulative coupling of aminopyridines with alkynes†

Yechan Kimab  and  Sungwoo Hong*ab  

* Corresponding authors

a Department of Chemistry, Korea Advanced Institute of Science and Technology (KAIST), Daejeon, Korea
E-mail: hongorg@kaist.ac.kr

b Center for Catalytic Hydrocarbon Functionalizations, Institute for Basic Science (IBS), Daejeon 305-701, Korea
Fax: +82-42-350-2810
Tel: +82-42-350-2811

Abstract

An efficient Rh(III)-catalyzed 7-azaindole synthesis was developed via C–H activation/annulative coupling of aminopyridines with alkynes. The reaction was highly regioselective and tolerated various functional groups, permitting the construction of various 7-azaindoles.

Graphical abstract: Rh(iii)-catalyzed 7-azaindole synthesis via C–H activation/annulative coupling of aminopyridines with alkynes

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Article information

DOI
https://doi.org/10.1039/C5CC03497C
Article type
Communication
Submitted
27 Apr 2015
Accepted
03 Jun 2015
First published
03 Jun 2015

Chem. Commun., 2015,51, 11202-11205

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Rh(III)-catalyzed 7-azaindole synthesis via C–H activation/annulative coupling of aminopyridines with alkynes

Y. Kim and S. Hong, Chem. Commun., 2015, 51, 11202 DOI: 10.1039/C5CC03497C

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