Issue 10, 2016
From the journal:

Organic & Biomolecular Chemistry

Regioselective Ir(iii)-catalyzed C–H alkynylation directed by 7-azaindoles†

Bin Liu,a   Xin Wang,a   Zemei Ge*a  and  Runtao Li*a  

* Corresponding authors

a Skate Key Laboratory of Natural and Biomimetic Drugs, Peking University, Beijing 100191, China
E-mail: lirt@bjmu.edu.cn

Abstract

Herein we report a novel iridium(III)-catalyzed ortho-mono-alkynylation of 7-azaindoles under mild conditions. This approach provides a general and straightforward access to form novel 7-azaindole derivatives with ample substrate scope and broad group tolerance.

Graphical abstract: Regioselective Ir(iii)-catalyzed C–H alkynylation directed by 7-azaindoles

About
Cited by
Related
Download options Please wait...

Supplementary files

Article information

DOI
https://doi.org/10.1039/C6OB00179C
Article type
Paper
Submitted
21 Jan 2016
Accepted
08 Feb 2016
First published
09 Feb 2016

Org. Biomol. Chem., 2016,14, 2944-2949

Permissions

Request permissions

Regioselective Ir(III)-catalyzed C–H alkynylation directed by 7-azaindoles

B. Liu, X. Wang, Z. Ge and R. Li, Org. Biomol. Chem., 2016, 14, 2944 DOI: 10.1039/C6OB00179C

To request permission to reproduce material from this article, please go to the Copyright Clearance Center request page.

If you are an author contributing to an RSC publication, you do not need to request permission provided correct acknowledgement is given.

If you are the author of this article, you do not need to request permission to reproduce figures and diagrams provided correct acknowledgement is given. If you want to reproduce the whole article in a third-party publication (excluding your thesis/dissertation for which permission is not required) please go to the Copyright Clearance Center request page.

Read more about how to correctly acknowledge RSC content.

Social activity

Spotlight

Advertisements